Emkhakheni wamakhemikhali wezokwelapha, amakhompiyutha ambalwa avelele ukusetshenziswa kwawo okuhlukahlukene kanye nokusebenza ngempumelelo njengeDibenzaberone. Le nhlanganisela eyingqayizivele, eyaziwa nangokuthi yi-1011-dihydrodibenza [A, D] cyclohepten-5-eyodwa, idonsele ukunakwa ngamandla alo okulapha emikhakheni ehlukahlukene yezokwelapha. Ake sithambeke ngokujulile emhlabeni weDibenzosuberone futhi sihlole izinzuzo zayo ukuze zibe yingxenye ebalulekile yezempilo yanamuhla.
Ngaphambili kocwaningo lwezokwelapha, iDibenzaberone imibukiso ekhombisa izakhiwo ezikhulisa inani layo. Kuyaziwa ngekhono layo lokusebenza njenge-prodrug, okusho ukuthi kungaguqulwa kube ama-ejenti asebenzayo emithi emzimbeni. Le mpahla eyingqayizivele inika amandla imiphumela yokwelapha ehambelana nezokwelapha ngenkathi inciphisa imiphumela emibi, okwenza kube ukukhetha kokuqala kwezidakamizwa.
Izicelo zokwelapha ze-Dibenzocycloconone zibanzi kakhulu futhi zibeke imikhakha eminingi yezokwelapha. Okubaluleke kakhulu kwalokhu kuyindima yayo ekwelapheni ukuphazamiseka kwe-neurological. Ucwaningo lukhombisa ukuthi i-Dibenzosuberone ingasiza ukudambisa izimpawu ezihambisana nezimo ezifana nesifo sikaParkinson, futhi kungasiza ekuqondisweni kweDopamine. Ngokwengeziwe, izakhiwo zayo ezingaba khona ezingaba khona ziye zahlolwa, ziphakamisa ukuthi zisetshenziswe ekwelashweni kwe-epilepsy.
Ngaphezu kwalokho, imiphumela elwa nokuvuvukala kwe-Dibenzosubeberone ifundelwe kakhulu, ivulwe ukuthi kungenzeka ukusetshenziswa kwayo ekwelapheni izifo ezivuthayo. Ukusuka ku-arthritis kuya ezifweni ze-autoimmune, leli khono le-compleate yokushintsha izimpendulo zokuzivikela komzimba lingaholela ekuthuthukisweni kokwelashwa okukhulu.
Ngaphezu kwalokhu, iDibenzaberone futhi isebenzisa futhi ku-endocrinology. Amandla awo okusebenzisana nohlelo lwe-hormonal lomzimba libonisa ukuthi lidlala indima ekunikezelweni kwezinqubo ezifana ne-metabolism ne-homeostasis yamandla. Lolu hlu olubanzi lwemisebenzi lukhombisa ukuguquguquka okuhlukahlukene nokubaluleka kwe-Dibenzosuberone kumakhemikhali okwelapha okwelapha.
Izinzuzo zeDibenzoCycloconone zandise ngaphezu kwemiphumela yayo yokwelapha. Isakhiwo saso samakhemikhali siguqulwa kalula, okuvumela abaphenyi ukuthi bathuthukise ukusulwa ngempumelelo noma imiphumela eqondisiwe. Lokhu kuvumelana nezimo ekwakheni nasekusetshenzisweni kwenza kube yithuluzi elibalulekile ekutholweni kwezidakamizwa nentuthuko.
Kulabo abafuna i-DibenzocyCloheptone ephezulu, iJingye Pharmaceutical inikeza izixazululo ezithembekile. Iwebhusayithi yabo ku-https://www.jingyepharma.com/dibenzosuberone-011-dihadibenzoadcyclohepten-5-one-product/Inikeza imininingwane ephelele ngale nhlanganisela eyenziwe ngezithonjana. UJingye Pharmaceuticals uzibophezele ebuhleni obuhle futhi unomlando wokukhiqiza amakhambi aphezulu, ukuqinisekisa ukuthi unokufinyelela okulula futhi okuthembekile eDibenzocyClohepTone.
Ngamafuphi, iDibenzaberone ikhombisa ukuthuthuka okusha kwisayensi yezemithi. Uhla lwayo olubanzi lwezicelo, kusuka ku-neurology ku-endocrinology, futhi amandla alo enziwe ngezifiso akwenze kube yitshe lezokwelapha lanamuhla. Njengoba siqhubeka nokuhlola ukujula kwalesi sakhiwo esimangalisayo, izinzuzo zeDibenzaberone ngokungangabazeki zizobumba ikusasa eliqhakazile ekunakekelweni kwezempilo.
VakashelaJingyeIzemithi namuhla ukuze ufunde kabanzi ngenqubekela phambili ye-Dreakthrough eyenziwe eDibenzaberone futhi ufunde ukuthi le nhlanganisela ingaguqula kanjani ukuqonda kwakho okusha kwezemithi.
Isikhathi sePosi: Mar-29-2024