Umenzi othembekile

Jiangsu jingye Pharmaceutical Co, Ltd.
Ikhasi_Banjaneri

Izindaba

Izicelo zezokwelapha zeDibenzosuberone

I-Dibenzosuberone, i-polycyclic aphungekile hydrocarbon, igxile kakhulu emphakathini wesayensi ngenxa yemisebenzi yayo yemvelo ethembisayo. Ngenkathi ikakhulukazi yaziwa ngendima yayo njengommeleli wokuhlanganiswa kwe-organic, iDibenzosuberone kanye nezinto zayo zokususelwa kwayo zikhombise amathuba okusetshenziswa okuhlukahlukene kwezokwelapha. Kulesi sihloko, sizohlola izinzuzo ezingaba khona kanye nokusetshenziswa kweDibenzosuberone emkhakheni wezokwelapha.

Izicelo zezokwelapha ezingaba khona

Izakhiwo ze-Anti-Cancer:

Izifundo eziningana ziveze ukuthi iDibenzosuberone kanye nezinto zalo zokususelwa kwayo zibonisa izakhiwo ezilwa nomdlavuza. Lezi zinhlanganisela zikhonjiswe ukuheha i-apoptosis (ukushona kwamaseli ahlelwe) kumaseli womdlavuza, kuvimbela ukukhula kwesikhukhula, futhi kuvikele i-metastasis.

Lezi zinqubo ezingaphansi kwale miphumela ziyinkimbinkimbi futhi zivame ukubandakanya ukuxhumana ngezindlela zokusayina amaselula.

Imiphumela ye-NeuroProtatect:

I-Dibenzosuberone ikhombisile imiphumela emihle ezifundweni zemvelo. Kukhonjiswe ukwehlisa ukucindezelwa okuyi-oxidative, ukuvuvukala, kanye nomonakalo we-neuronal obangelwa ukuphazamiseka okuhlukahlukene kwemizwa.

Le mpikiswano inganikeza izinzuzo ezingaba khona zokwelapha ezingaba yizimo ezifana nesifo se-Alzheimer's, isifo sikaParkinson, kanye noStroke.

Umsebenzi wokulwa nokuvuvukala:

I-Dibenzosuberone ibonise izakhiwo zokulwa nokuvuvukala, okwenza kube ngumuntu ongabenza abe ngumele imali yokwelashwa kwezifo ezivuthayo. Kungasiza ukunciphisa ukuvuvukala ngokuvimbela ukukhiqizwa kwama-cytokines okuvuvukala.

Umsebenzi we-antimicrobial:

Okunye okuvela kokutholwa kweDibenzosuberone kukhombise umsebenzi wokulwa namagciwane abhekene nohla lwamagciwane nesikhunta. Le mpahla ingabenza balusizo ekuthuthukisweni kwama-antibiotic amasha nama-antifungal agents.

Izindlela zokusebenza

Izindlela eziqondile lapho uDibenzosuberone esebenzisa khona imiphumela yalo yemvelo aziqondakali ngokuphelele kepha kucatshangwa ukuthi zibandakanya ukusebenzisana nokuhlosiwe okuhlukahlukene kwamaselula, kufaka phakathi:

Ama-receptors: I-Dibenzosuberone ingabopha futhi isebenze noma ivimbele ama-receptors athile, okuholela emicimbini yokusayina ephansi.

Ama-enzyme: Le mpikiswano ingavimba noma isebenze ama-enzyme athile athinteka ezinqubweni zamaselula anjengesakhiwo semali yeseli, i-apoptosis, kanye nokuvuvukala.

Ukuxineka nge-oxidative: I-Dibenzosuberone ingasebenza njenge-antioxidant, ukuvikela amaseli emmowazini odalwe izinhlobo ze-oksijini ezisebenzayo.

Izinselelo nezinkomba zesikhathi esizayo

Ngenkathi ukusetshenziswa kwezokwelapha okungaba khona kweDibenzosuberone kuyathembisa, kunezingqinamba eziningana ezidinga ukubhekelwa ngaphambi kokuthi zisetshenziswe njenge-ejenti yokwelapha. Lokhu kufaka phakathi:

Ubuthi: Ubuthi beDibenzosuberone kanye nezinto zokutholwa kwalo kumele kuhlolwe ngokucophelela ukuze kuqinisekiswe ukuphepha kwabo ekusetshenzisweni komuntu.

I-Bioavailability: Ukuthuthukisa i-Bioavailability yeDibenzaberone kubalulekile ukulethwa kwayo okusebenzayo ekuhlose izicubu.

Ukwakhiwa kwezidakamizwa: Ukuthuthukisa ukwakhiwa kwezidakamizwa okufanelekile kokulethwa kweDibenzosuberone kuwumsebenzi oyinkimbinkimbi.

Ukugcina

I-Dibenzosuberone kanye nokutholwa kwayo kubonisa indawo ethembisayo yocwaningo ngezinhlelo zokusebenza ezingaba khona ekwelapheni izifo ezahlukahlukene. Ezinye izifundo ziyadingeka ukuqonda izindlela zokusebenza kwalezi zinhlaka kanye nokuthuthukisa abenzeli abaphephile nabasebenzayo.


Isikhathi sePosi: Aug-29-2024